The antimalarial drug mefloquine enhances TP53 premature termination codon readthrough by aminoglycoside G418 MW Ferguson, CAN Gerak, CCT Chow, EJ Rastelli, KE Elmore, F Stahl, ... PLoS One 14 (5), e0216423, 2019 | 26 | 2019 |
The role of silk in courtship and chemical communication of the false widow spider, Steatoda grossa (Araneae: Theridiidae) C Scott, C Gerak, S McCann, G Gries Journal of ethology 36, 191-197, 2018 | 17 | 2018 |
Both chemical and non-chemical steps limit the catalytic efficiency of family 4 glycoside hydrolases N Sannikova, CAN Gerak, FS Shidmoossavee, DT King, ... Biochemistry 57 (24), 3378-3386, 2018 | 9 | 2018 |
Biophysical characterization of the ETV6 PNT domain polymerization interfaces CAN Gerak, SY Cho, M Kolesnikov, M Okon, MEP Murphy, RB Sessions, ... Journal of Biological Chemistry 296, 2021 | 4 | 2021 |
A biosensor of protein foldedness identifies increased “holdase” activity of chaperones in the nucleus following increased cytosolic protein aggregation CB Raeburn, AR Ormsby, D Cox, CA Gerak, C Makhoul, NS Moily, ... Journal of Biological Chemistry 298 (8), 2022 | 3 | 2022 |
A multipronged screening approach targeting inhibition of ETV6 PNT domain polymerization CAN Gerak, SM Zhang, AD Balgi, IJ Sadowski, RB Sessions, LP McIntosh, ... SLAS DISCOVERY: Advancing the Science of Drug Discovery 26 (5), 698-711, 2021 | 2 | 2021 |
Insights into the inhibition of ETV6 PNT domain polymerization CAN Gerak University of British Columbia, 2020 | 1 | 2020 |
WANTED: SMALL MOLECULES TO INHIBIT PNT DOMAIN-MEDIATED POLYMERIZATION OF ETV6 CHIMERIC ONCOPROTEINS C Gerak, S Cho, M Okon, R Sessions, M Roberge, L McIntosh PROTEIN SCIENCE 28, 48-48, 2019 | | 2019 |
IDENTIFYING HOT SPOT RESIDUES AT THE ETV6 PNT DOMAIN POLYMERIZATION INTERFACE S Cho, C Gerak, M Roberge, L McIntosh PROTEIN SCIENCE 28, 148-148, 2019 | | 2019 |