Folgen
Ghotas Evindar
Ghotas Evindar
Bestätigte E-Mail-Adresse bei gsk.com - Startseite
Titel
Zitiert von
Zitiert von
Jahr
Parallel Synthesis of a Library of Benzoxazoles and Benzothiazoles Using Ligand-Accelerated Copper-Catalyzed Cyclizations of ortho-Halobenzanilides
G Evindar, RA Batey
The Journal of Organic Chemistry 71 (5), 1802-1808, 2006
6282006
Copper-catalyzed domino annulation approaches to the synthesis of benzoxazoles under microwave-accelerated and conventional thermal conditions
RD Viirre, G Evindar, RA Batey
The Journal of organic chemistry 73 (9), 3452-3459, 2008
3092008
Copper-and palladium-catalyzed intramolecular aryl guanidinylation: an efficient method for the synthesis of 2-aminobenzimidazoles
G Evindar, RA Batey
Organic Letters 5 (2), 133-136, 2003
2802003
Discovery of Thieno[3,2-d]pyrimidine-6-carboxamides as Potent Inhibitors of SIRT1, SIRT2, and SIRT3
JS Disch, G Evindar, CH Chiu, CA Blum, H Dai, L Jin, E Schuman, ...
Journal of medicinal chemistry 56 (9), 3666-3679, 2013
2052013
Copper-and palladium-catalyzed intramolecular C–S bond formation: a convenient synthesis of 2-aminobenzothiazoles
LL Joyce, G Evindar, RA Batey
Chemical communications, 446-447, 2004
1252004
Encoded library technology as a source of hits for the discovery and lead optimization of a potent and selective class of bactericidal direct inhibitors of Mycobacterium …
L Encinas, H O’Keefe, M Neu, MJ Remuiñán, AM Patel, A Guardia, ...
Journal of Medicinal Chemistry 57 (4), 1276-1288, 2014
1202014
Stereoselective synthesis of threo and erythro β-hydroxy and β-disubstituted-β-hydroxy α-amino acids
MA Blaskovich, G Evindar, NGW Rose, S Wilkinson, Y Luo, GA Lajoie
The Journal of Organic Chemistry 63 (11), 3631-3646, 1998
1161998
Application of encoded library technology (ELT) to a protein–protein interaction target: Discovery of a potent class of integrin lymphocyte function-associated antigen 1 (LFA-1 …
CS Kollmann, X Bai, CH Tsai, H Yang, KE Lind, SR Skinner, Z Zhu, ...
Bioorganic & Medicinal Chemistry 22 (7), 2353-2365, 2014
962014
Design and application of a DNA-encoded macrocyclic peptide library
Z Zhu, A Shaginian, LSC Grady, T O’Keeffe, XE Shi, CP Davie, ...
ACS Chemical Biology 13 (1), 53-59, 2018
922018
The discovery of VX-745: A novel and selective p38α kinase inhibitor
JP Duffy, EM Harrington, FG Salituro, JE Cochran, J Green, H Gao, ...
ACS Medicinal Chemistry Letters 2 (10), 758-763, 2011
882011
Discovery of a potent class of PI3Kα inhibitors with unique binding mode via encoded library technology (ELT)
H Yang, PF Medeiros, K Raha, P Elkins, KE Lind, R Lehr, ND Adams, ...
ACS medicinal chemistry letters 6 (5), 531-536, 2015
712015
Prioritizing multiple therapeutic targets in parallel using automated DNA-encoded library screening
CA Machutta, CS Kollmann, KE Lind, X Bai, PF Chan, J Huang, L Ballell, ...
Nature communications 8 (1), 16081, 2017
702017
DNA-encoded library technology-based discovery, lead optimization, and prodrug strategy toward structurally unique indoleamine 2, 3-dioxygenase-1 (IDO1) Inhibitors
WM Kazmierski, B Xia, J Miller, M De la Rosa, D Favre, RM Dunham, ...
Journal of Medicinal Chemistry 63 (7), 3552-3562, 2020
532020
Methods and compositions for modulating sphingosine-1-phosphate (S1P) receptor activity
G Evindar, H Deng, B Morgan
US Patent App. 11/349,069, 2006
382006
Discovery and characterization of a class of pyrazole inhibitors of bacterial undecaprenyl pyrophosphate synthase
N Concha, J Huang, X Bai, A Benowitz, P Brady, LSC Grady, LH Kryn, ...
Journal of Medicinal Chemistry 59 (15), 7299-7304, 2016
372016
Methods and compositions for modulating sphingosine-1-phosphate (S1P) receptor activity
AK Saha, MJ Kavarana, G Evindar, AL Satz, B Morgan
US Patent 7,241,812, 2007
362007
Methods and compositions for modulating sphingosine-1-phosphate (S1P) receptor activity
AK Saha, MJ Kavarana, G Evindar, AL Satz, B Morgan
US Patent 7,241,812, 2007
362007
Peptide heterocycle conjugates: A diverted Edman degradation protocol for the synthesis of N-terminal 2-iminohydantoins
G Evindar, RA Batey
Organic Letters 5 (8), 1201-1204, 2003
362003
Inhibitors of p38
F Salituro, G Bemis, H Gao, G Evindar
US Patent 6,635,644, 2003
352003
Recent developments in the synthesis of nitrogen-containing heterocycles through C–H/N–h bond functionalizations and oxidative cyclization
X Liu, Y Huang, X Meng, J Li, D Wang, Y Chen, D Tang, B Chen
Synlett 30 (09), 1026-1036, 2019
322019
Das System kann den Vorgang jetzt nicht ausführen. Versuchen Sie es später erneut.
Artikel 1–20