Discovery of tropinone-thiazole derivatives as potent caspase 3/7 activators, and noncompetitive tyrosinase inhibitors with high antiproliferative activity: Rational design … K Piechowska, M Świtalska, J Cytarska, K Jaroch, K Łuczykowski, ... European journal of medicinal chemistry 175, 162-171, 2019 | 43 | 2019 |
Synthesis, antimicrobial activity, and determination of the lipophilicity of ((cyclohex-3-enylmethylene) hydrazinyl) thiazole derivatives A Biernasiuk, M Kawczyńska, A Berecka-Rycerz, B Rosada, ... Medicinal Chemistry Research 28, 2023-2036, 2019 | 35 | 2019 |
Synthesis, antimicrobial evaluation and theoretical prediction of NMR chemical shifts of thiazole and selenazole derivatives with high antifungal activity against Candida spp. KZ Łączkowski, K Motylewska, A Baranowska-Łączkowska, A Biernasiuk, ... Journal of Molecular Structure 1108, 427-437, 2016 | 34 | 2016 |
Synthesis and in vitro antiproliferative activity of thiazole-based nitrogen mustards: the hydrogen bonding interaction between model systems and nucleobases K Z Laczkowski, K Misiura, M Switalska, J Wietrzyk, ... Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2014 | 32 | 2014 |
Benzo [b] thiophene-thiazoles as potent anti-Toxoplasma gondii agents: Design, synthesis, tyrosinase/tyrosine hydroxylase inhibitors, molecular docking study, and antioxidant … B Rosada, A Bekier, J Cytarska, W Płaziński, O Zavyalova, A Sikora, ... European Journal of Medicinal Chemistry 184, 111765, 2019 | 31 | 2019 |
Thiazoles with cyclopropyl fragment as antifungal, anticonvulsant, and anti-Toxoplasma gondii agents: synthesis, toxicity evaluation, and molecular docking study KZ Łączkowski, N Konklewska, A Biernasiuk, A Malm, K Sałat, A Furgała, ... Medicinal Chemistry Research 27, 2125-2140, 2018 | 31 | 2018 |
Synthesis, antimicrobial and anticonvulsant screening of small library of tetrahydro-2H-thiopyran-4-yl based thiazoles and selenazoles KZ Łączkowski, A Biernasiuk, A Baranowska-Łączkowska, S Zielińska, ... Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup2), 24-39, 2016 | 31 | 2016 |
Synthesis and anticonvulsant activities of novel 2-(cyclopentylmethylene) hydrazinyl-1, 3-thiazoles in mouse models of seizures KZ Łączkowski, K Sałat, K Misiura, A Podkowa, N Malikowska Journal of Enzyme Inhibition and Medicinal Chemistry 31 (6), 1576-1582, 2016 | 30 | 2016 |
The newly synthesized thiazole derivatives as potential antifungal compounds against Candida albicans A Biernasiuk, A Berecka-Rycerz, A Gumieniczek, M Malm, KZ Łączkowski, ... Applied Microbiology and Biotechnology 105 (16), 6355-6367, 2021 | 29 | 2021 |
Synthesis, in vitro biological screening and molecular docking studies of novel camphor-based thiazoles K Z Laczkowski, K Misiura, A Biernasiuk, A Malm, A Siwek, T Plech, ... Medicinal Chemistry 10 (6), 600-608, 2014 | 29 | 2014 |
The ORP basis set designed for optical rotation calculations A Baranowska‐Łączkowska, KZ Łączkowski Journal of Computational Chemistry 34 (23), 2006-2013, 2013 | 29 | 2013 |
Model studies of the optical rotation, and theoretical determination of its sign for β‐pinene and trans‐pinane A Baranowska, KZ Ła̧czkowski, AJ Sadlej Journal of computational chemistry 31 (6), 1176-1181, 2010 | 29 | 2010 |
One-pot telescoped synthesis of thiazole derivatives from β-keto esters and thioureas promoted by tribromoisocyanuric acid VSC de Andrade, MCS de Mattos Synthesis 50 (24), 4867-4874, 2018 | 26 | 2018 |
Thiazole-based nitrogen mustards: design, synthesis, spectroscopic studies, DFT calculation, molecular docking, and antiproliferative activity against selected human cancer … KZ Łączkowski, M Świtalska, A Baranowska-Łączkowska, T Plech, ... Journal of Molecular Structure 1119, 139-150, 2016 | 26 | 2016 |
Synthesis, molecular docking, ctDNA interaction, DFT calculation and evaluation of antiproliferative and anti-Toxoplasma gondii activities of 2,4-diaminotriazine … KZ Łączkowski, J Anusiak, M Świtalska, K Dzitko, J Cytarska, ... Medicinal Chemistry Research 27, 1131-1148, 2018 | 25 | 2018 |
Effect of the dichloro-substitution on antiproliferative activity of phthalimide-thiazole derivatives. Rational design, synthesis, elastase, caspase 3/7, and EGFR tyrosine … B Donarska, M Świtalska, W Płaziński, J Wietrzyk, KZ Łączkowski Bioorganic Chemistry 110, 104819, 2021 | 24 | 2021 |
Tropinone-derived alkaloids as potent anticancer agents: Synthesis, tyrosinase inhibition, mechanism of action, DFT calculation, and molecular docking studies K Piechowska, M Mizerska-Kowalska, B Zdzisińska, J Cytarska, ... International Journal of Molecular Sciences 21 (23), 9050, 2020 | 18 | 2020 |
Asymmetric synthesis of N-substituted N-hydroxyureas KZ Łączkowski, MM Pakulski, MP Krzemiński, P Jaisankar, M Zaidlewicz Tetrahedron: Asymmetry 19 (7), 788-795, 2008 | 18 | 2008 |
Antibacterial Activity, Interaction with Nucleobase and Molecular Docking Studies of 4-Formylbenzoic Acid Based Thiazoles KZ Łączkowski, A Biernasiuk, A Baranowska-Łączkowska, et al. Medicinal Chemistry 12, 553-562, 2016 | 16* | 2016 |
Synthesis, antimicrobial activities and molecular docking studies of novel 6-hydroxybenzofuran-3 (2H)-one based 2, 4-disubstituted 1, 3-thiazoles K Z Laczkowski, K Misiura, A Biernasiuk, A Malm, A Siwek, T Plech Letters in Drug Design & Discovery 10 (9), 798-807, 2013 | 16 | 2013 |