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Lindsey Burggraaff
Lindsey Burggraaff
Verified email at lacdr.leidenuniv.nl
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Year
Advances and challenges in computational target prediction
D Sydow, L Burggraaff, A Szengel, HWT van Vlijmen, AP IJzerman, ...
Journal of chemical information and modeling 59 (5), 1728-1742, 2019
972019
Activity-based protein profiling identifies α-ketoamides as inhibitors for phospholipase A2 group XVI
J Zhou, ED Mock, A Martella, V Kantae, X Di, L Burggraaff, MP Baggelaar, ...
ACS Chemical Biology 14 (2), 164-169, 2019
292019
Identification of novel small molecule inhibitors for solute carrier SGLT1 using proteochemometric modeling
L Burggraaff, P Oranje, R Gouka, P van der Pijl, M Geldof, ...
Journal of cheminformatics 11, 1-10, 2019
252019
Development of ubiquitin‐based probe for metalloprotease deubiquitinases
DS Hameed, A Sapmaz, L Burggraaff, A Amore, CJ Slingerland, ...
Angewandte Chemie International Edition 58 (41), 14477-14482, 2019
232019
Rapid screening and identification of ACE inhibitors in snake venoms using at-line nanofractionation LC-MS
M Mladic, T de Waal, L Burggraaff, J Slagboom, GW Somsen, ...
Analytical and bioanalytical chemistry 409, 5987-5997, 2017
222017
Novel natural and synthetic inhibitors of solute carriers SGLT1 and SGLT2
P Oranje, R Gouka, L Burggraaff, M Vermeer, C Chalet, G Duchateau, ...
Pharmacology Research & Perspectives 7 (4), e00504, 2019
212019
Development of a retinal-based probe for the profiling of retinaldehyde dehydrogenases in cancer cells
STA Koenders, LS Wijaya, MN Erkelens, AT Bakker, VE van der Noord, ...
ACS central science 5 (12), 1965-1974, 2019
172019
Quantitative prediction of selectivity between the A1 and A2A adenosine receptors
L Burggraaff, HWT van Vlijmen, AP IJzerman, GJP van Westen
Journal of Cheminformatics 12, 1-16, 2020
132020
Design and pharmacological profile of a novel covalent partial agonist for the adenosine A1 receptor
X Yang, MA Dilweg, D Osemwengie, L Burggraaff, D van der Es, ...
Biochemical Pharmacology 180, 114144, 2020
132020
Structure–activity relationship studies of α-ketoamides as inhibitors of the phospholipase A and acyltransferase enzyme family
J Zhou, ED Mock, K Al Ayed, X Di, V Kantae, L Burggraaff, AF Stevens, ...
Journal of Medicinal Chemistry 63 (17), 9340-9359, 2020
122020
Identification of novel small molecule inhibitors for solute carrier SGLT1 using proteochemometric modeling. J Cheminform 11: 15
L Burggraaff, P Oranje, R Gouka, P Van Der Pijl, M Geldof, ...
62019
Successive statistical and structure-based modeling to identify chemically novel kinase inhibitors
L Burggraaff, EB Lenselink, W Jespers, J van Engelen, BJ Bongers, ...
Journal of Chemical Information and Modeling 60 (9), 4283-4295, 2020
52020
Annotation of allosteric compounds to enhance bioactivity modeling for class a GPCRs
L Burggraaff, A van Veen, CC Lam, HWT van Vlijmen, AP IJzerman, ...
Journal of Chemical Information and Modeling 60 (10), 4664-4672, 2020
32020
A multiple classifier system identifies novel cannabinoid CB2 receptor ligands
D Ruano-Ordás, L Burggraaff, R Liu, C van der Horst, LH Heitman, ...
Journal of Cheminformatics 11, 1-14, 2019
32019
Synthesis and SAR evaluation of coumarin derivatives as potent cannabinoid receptor agonists
F Mohr, T Hurrle, L Burggraaff, L Langer, MP Bemelmans, M Knab, ...
European Journal of Medicinal Chemistry 220, 113354, 2021
22021
Proteins in harmony: Tuning selectivity in early drug discovery
L Burggraaff
Leiden University, 2020
2020
Design, Synthesis and Pharmacological Profile of LUF7746, a Novel Covalent Partial Agonist for the Adenosine A1 Receptor
X Yang, M Dilweg, D Osemwengie, L Burggraaff, D van der Es, L Heitman, ...
2020
Quantitative prediction of selectivity between the A
L Burggraaff, HWT van Vlijmen, AP IJzerman, GJP van Westen
2020
Chapter two Advances and Challenges in Computational Target Prediction
D Sydow, L Burggraaff, A Szengel, HWT van Vlijmen, AP IJzerman, ...
Proteins in Harmony Tuning Selectivity in Early Drug Discovery, 21, 0
Chapter three Identification of Novel Small Molecule Inhibitors for Solute Carrier SGLT1 using Proteochemometric Modeling
L Burggraaff, P Oranje, R Gouka, P van der Pijl, M Geldof, H WT
Proteins in Harmony Tuning Selectivity in Early Drug Discovery, 49, 0
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Articles 1–20