Pancreatic lipase inhibition activity of trilactone terpenes of Ginkgo biloba Y Bustanji, IM Al-Masri, M Mohammad, M Hudaib, K Tawaha, H Tarazi, ... Journal of Enzyme Inhibition and Medicinal Chemistry 26 (4), 453-459, 2011 | 123 | 2011 |
Safranal induces DNA double-strand breakage and ER-stress-mediated cell death in hepatocellular carcinoma cells A Al-Hrout, A Chaiboonchoe, B Khraiwesh, C Murali, B Baig, R El-Awady, ... Scientific reports 8 (1), 16951, 2018 | 99 | 2018 |
Camel whey protein hydrolysates induced G2/M cellcycle arrest in human colorectal carcinoma C Murali, P Mudgil, CY Gan, H Tarazi, R El-Awady, Y Abdalla, A Amin, ... Scientific reports 11 (1), 7062, 2021 | 48 | 2021 |
A review of HER4 (ErbB4) kinase, its impact on cancer, and its inhibitors MI El-Gamal, NH Mewafi, NE Abdelmotteleb, MA Emara, H Tarazi, ... Molecules 26 (23), 7376, 2021 | 36 | 2021 |
Post-Ugi cascade transformations for accessing diverse chromenopyrrole collections V Srinivasulu, SMN Sieburth, R El-Awady, NM Kariem, H Tarazi, ... Organic letters 20 (3), 836-839, 2018 | 36 | 2018 |
Rational design, synthesis, pharmacophore modeling, and docking studies for identification of novel potent DNA-PK inhibitors S Ihmaid, HEA Ahmed, AAS Ali, YE Sherif, HM Tarazi, SM Riyadh, ... Bioorganic Chemistry 72, 234-247, 2017 | 35 | 2017 |
Inhibition of SHP2 by new compounds induces differential effects on RAS/RAF/ERK and PI3K/AKT pathways in different cancer cell types CG Vazhappilly, E Saleh, W Ramadan, V Menon, AM Al-Azawi, H Tarazi, ... Investigational new drugs 37, 252-261, 2019 | 33 | 2019 |
Design, synthesis and SAR analysis of potent BACE1 inhibitors: Possible lead drug candidates for Alzheimer's disease H Tarazi, RA Odeh, R Al-Qawasmeh, IA Yousef, W Voelter, TH Al-Tel European Journal of Medicinal Chemistry 125, 1213-1224, 2017 | 32 | 2017 |
One-pot synthesis of diverse collections of benzoxazepine and indolopyrazine fused to heterocyclic systems V Srinivasulu, I Shehadeh, MA Khanfar, OG Malik, H Tarazi, ... The Journal of Organic Chemistry 84 (2), 934-948, 2018 | 27 | 2018 |
An Efficient Synthesis of bi‐Aryl Pyrimidine Heterocycles: Potential New Drug Candidates to Treat Alzheimer's Disease TU Rehman, IU Khan, M Ashraf, H Tarazi, S Riaz, M Yar Archiv der Pharmazie 350 (3-4), 1600304, 2017 | 25 | 2017 |
Design and synthesis of new RAF kinase-inhibiting antiproliferative quinoline derivatives. Part 2: Diarylurea derivatives MI El-Gamal, MA Khan, H Tarazi, MS Abdel-Maksoud, MMG El-Din, ... European Journal of Medicinal Chemistry 127, 413-423, 2017 | 24 | 2017 |
Current status of baricitinib as a repurposed therapy for COVID-19 M Saber-Ayad, S Hammoudeh, E Abu-Gharbieh, R Hamoudi, H Tarazi, ... Pharmaceuticals 14 (7), 680, 2021 | 22 | 2021 |
Design, synthesis and biological evaluation of new pyrrolidine carboxamide analogues as potential chemotherapeutic agents for hepatocellular carcinoma HA Omar, DM Zaher, V Srinivasulu, F Hersi, H Tarazi, TH Al-Tel European Journal of Medicinal Chemistry 139, 804-814, 2017 | 22 | 2017 |
Imidazothiazole-based potent inhibitors of V600E-B-RAF kinase with promising anti-melanoma activity: Biological and computational studies HS Anbar, MI El-Gamal, H Tarazi, BS Lee, HR Jeon, D Kwon, CH Oh Journal of Enzyme Inhibition and Medicinal Chemistry 35 (1), 1712-1726, 2020 | 18 | 2020 |
Discovery of first-in-class imidazothiazole-based potent and selective ErbB4 (HER4) kinase inhibitors SO Zaraei, RM Sbenati, NN Alach, HS Anbar, R El-Gamal, H Tarazi, ... European Journal of Medicinal Chemistry 224, 113674, 2021 | 17 | 2021 |
Hepatoprotective and antioxidant potential of Nyctanthes arbor-tristis L. leaves against antitubercular drugs induced hepatotoxicity S Chaudhary, RK Gupta, A Kumar, H Tarazi Journal of Pharmacy & Pharmacognosy Research 6 (3), 205-215, 2018 | 17 | 2018 |
Enhancing student communication skills through Arabic language competency and simulated patient assessments S Hasan, DAH Hilal American Journal of Pharmaceutical Education 81 (4), 76, 2017 | 17 | 2017 |
Discovery of novel small-molecule inhibitors of SARS-CoV-2 main protease as potential leads for COVID-19 treatment A Manandhar, V Srinivasulu, M Hamad, H Tarazi, H Omar, DJ Colussi, ... Journal of Chemical Information and Modeling 61 (9), 4745-4757, 2021 | 14 | 2021 |
Conjugation of 4-aminosalicylate with thiazolinones afforded non-cytotoxic potent in vitro and in vivo anti-inflammatory hybrids HHM Abdu-Allah, AAB Abdelmoez, H Tarazi, ANA El-Shorbagi, ... Bioorganic Chemistry 94, 103378, 2020 | 14 | 2020 |
Bis-(5-substituted-2-thiono-1, 3, 5-thiadiazinan-3-yl) butane as a scaffold of anti-proliferative activity, blended by a multicomponent process AN El-Shorbagi, M El-Naggar, H Tarazi, S Chaudhary, H Abdu-Allah, ... Medicinal Chemistry Research 27, 1103-1110, 2018 | 14 | 2018 |