Bikash Debnath
Bikash Debnath
Assistant Research Scientist
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Cited by
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Role of the CXCL8-CXCR1/2 axis in cancer and inflammatory diseases
H Ha, B Debnath, N Neamati
Theranostics 7 (6), 1543, 2017
Small molecule inhibitors of CXCR4
B Debnath, S Xu, F Grande, A Garofalo, N Neamati
Theranostics 3 (1), 47, 2013
Discovery of an orally active small-molecule irreversible inhibitor of protein disulfide isomerase for ovarian cancer treatment
S Xu, AN Butkevich, R Yamada, Y Zhou, B Debnath, R Duncan, E Zandi, ...
Proceedings of the National Academy of Sciences 109 (40), 16348-16353, 2012
Small molecule inhibitors of signal transducer and activator of transcription 3 (Stat3) protein
B Debnath, S Xu, N Neamati
Journal of medicinal chemistry 55 (15), 6645-6668, 2012
Fragment-based discovery of 8-hydroxyquinoline inhibitors of the hiv-1 integrase–lens epithelium-derived growth factor/p75 (in–ledgf/p75) interaction
E Serrao, B Debnath, H Otake, Y Kuang, F Christ, Z Debyser, N Neamati
Journal of medicinal chemistry 56 (6), 2311-2322, 2013
Design of HIV-1 integrase inhibitors targeting the catalytic domain as well as its interaction with LEDGF/p75: a scaffold hopping approach using salicylate and catechol groups
X Fan, FH Zhang, RI Al-Safi, LF Zeng, Y Shabaik, B Debnath, ...
Bioorganic & medicinal chemistry 19 (16), 4935-4952, 2011
QSAR study on some pyridoacridine ascididemin analogues as anti-tumor agents
B Debnath, S Gayen, S Bhattacharya, S Samanta, T Jha
Bioorganic & medicinal chemistry 11 (24), 5493-5499, 2003
Discovery of a novel series of inhibitors of lymphoid tyrosine phosphatase with activity in human T cells
SM Stanford, D Krishnamurthy, MD Falk, R Messina, B Debnath, S Li, ...
Journal of medicinal chemistry 54 (6), 1640-1654, 2011
Repositioning HIV-1 integrase inhibitors for cancer therapeutics: 1, 6-naphthyridine-7-carboxamide as a promising scaffold with drug-like properties
LF Zeng, Y Wang, R Kazemi, S Xu, ZL Xu, TW Sanchez, LM Yang, ...
Journal of Medicinal Chemistry 55 (22), 9492-9509, 2012
5-N-Substituted-2-(substituted benzenesulphonyl) glutamines as antitumor agents. Part II: Synthesis, biological activity and QSAR study
S Samanta, K Srikanth, S Banerjee, B Debnath, S Gayen, T Jha
Bioorganic & medicinal chemistry 12 (6), 1413-1423, 2004
QSAR study on some anti-HIV HEPT analogues using physicochemical and topological parameters
S Gayen, B Debnath, S Samanta, T Jha
Bioorganic & medicinal chemistry 12 (6), 1493-1503, 2004
Structure-based optimization of a novel class of aldehyde dehydrogenase 1A (ALDH1A) subfamily-selective inhibitors as potential adjuncts to ovarian cancer chemotherapy
BC Huddle, E Grimley, CD Buchman, M Chtcherbinine, B Debnath, ...
Journal of medicinal chemistry 61 (19), 8754-8773, 2018
The Hydroxyquinoline Analogue YUM70 Inhibits GRP78 to Induce ER Stress–Mediated Apoptosis in Pancreatic Cancer
S Samanta, S Yang, B Debnath, D Xue, Y Kuang, K Ramkumar, AS Lee, ...
Cancer research 81 (7), 1883-1895, 2021
Discovery of a novel 5-carbonyl-1H-imidazole-4-carboxamide class of inhibitors of the HIV-1 integrase–LEDGF/p75 interaction
E Serrao, ZL Xu, B Debnath, F Christ, Z Debyser, YQ Long, N Neamati
Bioorganic & medicinal chemistry 21 (19), 5963-5972, 2013
Mechanistic evaluation and transcriptional signature of a glutathione S-transferase omega 1 inhibitor
K Ramkumar, S Samanta, A Kyani, S Yang, S Tamura, E Ziemke, ...
Nature communications 7 (1), 13084, 2016
Syntheses, biological evaluation and QSAR study on antitumor activity of 1, 5-N, N′-disubstituted-2-(substituted benzenesulphonyl) glutamamides
K Srikanth, B Debnath, T Jha
Bioorganic & medicinal chemistry 10 (6), 1841-1854, 2002
Synergistic effect of methanol extract of Abies webbiana leaves on sleeping time induced by standard sedatives in mice and anti-inflammatory activity of extracts in rats
SS Nayak, AK Ghosh, B Debnath, SP Vishnoi, T Jha
Journal of ethnopharmacology 93 (2-3), 397-402, 2004
QSAR study on some p-arylthio cinnamides as antagonists of biochemical ICAM-1/LFA-1 interaction and ICAM-1/JY-8 cell adhesion in relation to anti-inflammatory activity
B Debnath, S Samanta, K Roy, T Jha
Bioorganic & medicinal chemistry 11 (8), 1615-1619, 2003
1,5-N,N'-Disubstituted-2-(Substituted Benzenesulphonyl)glutamamides as Antitumor Agents. Part 2. Synthesis, Biological Activity and QSAR Study
B Debnath, K Srikanth, S Banarjee, T Jha
Internet Electronic Journal of Molecular Design 1 (10), 488-502, 2002
Exploring QSAR on 3-aminopyrazoles as antitumor agents for their inhibitory activity of CDK2/cyclin A
S Samanta, B Debnath, A Basu, S Gayen, K Srikanth, T Jha
European journal of medicinal chemistry 41 (10), 1190-1195, 2006
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