The 3F Library: Fluorinated Fsp3‐Rich Fragments for Expeditious 19F NMR Based Screening NS Troelsen, E Shanina, D Gonzalez‐Romero, D Danková, ISA Jensen, ... Angewandte Chemie 132 (6), 2224-2230, 2020 | 69 | 2020 |
Identification of multiple druggable secondary sites by fragment screening against DC‐SIGN J Aretz, H Baukmann, E Shanina, J Hanske, R Wawrzinek, VA Zapol'skii, ... Angewandte Chemie International Edition 56 (25), 7292-7296, 2017 | 47 | 2017 |
Stereoselective Synthesis of Fluorinated Galactopyranosides as Potential Molecular Probes for Galactophilic Proteins: Assessment of Monofluorogalactoside–LecA Interactions V Denavit, D Lainé, C Bouzriba, E Shanina, E Gillon, S Fortin, ... Chemistry–A European Journal 25 (17), 4478-4490, 2019 | 43 | 2019 |
Intradomain allosteric network modulates calcium affinity of the C-type lectin receptor langerin J Hanske, S Aleksić, M Ballaschk, M Jurk, E Shanina, M Beerbaum, ... Journal of the American Chemical Society 138 (37), 12176-12186, 2016 | 43 | 2016 |
Human CD22 inhibits murine B cell receptor activation in a human CD22 transgenic mouse model KJ Bednar, E Shanina, R Ballet, EP Connors, S Duan, J Juan, BM Arlian, ... The Journal of Immunology 199 (9), 3116-3128, 2017 | 36 | 2017 |
Automated Glycan Assembly of 19F‐labeled Glycan Probes Enables High‐Throughput NMR Studies of Protein–Glycan Interactions G Fittolani, E Shanina, M Guberman, PH Seeberger, C Rademacher, ... Angewandte Chemie International Edition 60 (24), 13302-13309, 2021 | 25 | 2021 |
Glycomimetics for the inhibition and modulation of lectins S Leusmann, P Ménová, E Shanin, A Titz, C Rademacher Chemical Society Reviews, 2023 | 22 | 2023 |
From pyrazolones to azaindoles: evolution of active-site SHP2 inhibitors based on scaffold hopping and bioisosteric replacement Y Mostinski, GJJE Heynen, MP López-Alberca, J Paul, S Miksche, ... Journal of medicinal chemistry 63 (23), 14780-14804, 2020 | 18 | 2020 |
Non‐carbohydrate glycomimetics as inhibitors of calcium (II)‐binding lectins S Kuhaudomlarp, E Siebs, E Shanina, J Topin, I Joachim, ... Angewandte Chemie 133 (15), 8185-8195, 2021 | 17 | 2021 |
Protein-observed 19F NMR of LecA from Pseudomonas aeruginosa E Shanina, E Siebs, H Zhang, D Varón Silva, I Joachim, A Titz, ... Glycobiology 31 (2), 159-165, 2021 | 16 | 2021 |
Targeting undruggable carbohydrate recognition sites through focused fragment library design E Shanina, S Kuhaudomlarp, E Siebs, FF Fuchsberger, M Denis, ... Communications Chemistry 5 (1), 64, 2022 | 9 | 2022 |
Targeting the Central Pocket of the Pseudomonas aeruginosa Lectin LecA E Siebs, E Shanina, S Kuhaudomlarp, ... ChemBioChem 23 (3), e202100563, 2022 | 9 | 2022 |
Druggable allosteric sites in β‐propeller lectins E Shanina, S Kuhaudomlarp, K Lal, PH Seeberger, A Imberty, ... Angewandte Chemie International Edition 61 (1), e202109339, 2022 | 9 | 2022 |
Identifikation sekundärer Bindestellen auf DC‐SIGN mithilfe eines Fragment‐Screenings J Aretz, H Baukmann, E Shanina, J Hanske, R Wawrzinek, VA Zapol'skii, ... Angewandte Chemie 129 (25), 7398-7402, 2017 | 8 | 2017 |
VA Zapol skii, PH Seeberger, DE Kaufmann, C. Rademacher J Aretz, H Baukmann, E Shanina, J Hanske, R Wawrzinek Angew. Chem. Int. Ed 56, 7292-7296, 2017 | 8 | 2017 |
Automatisierte Glykan‐Assemblierung 19F‐markierter Glykansonden ermöglicht Hochdurchsatz‐NMR‐Untersuchungen von Protein‐Glykan‐Interaktionen G Fittolani, E Shanina, M Guberman, PH Seeberger, C Rademacher, ... Angewandte Chemie 133 (24), 13414-13421, 2021 | 4 | 2021 |
Chemotherapy-induced, broadly reactive autoantibodies in a colon cancer patient F Broecker, E Shanin, N Lysov, V Shanin Cureus 14 (11), 2022 | 2 | 2022 |
Novel Chemotypes for Inhibition of Bacterial and Mammalian Carbohydrate-Binding Proteins E Shanina | | 2023 |
Allosterische, Wirkstoff‐zugängliche Bindestellen in β‐Propeller‐Lektinen E Shanina, S Kuhaudomlarp, K Lal, PH Seeberger, A Imberty, ... Angewandte Chemie 134 (1), e202109339, 2022 | | 2022 |
Stereoselective synthesis of fluorinated galactopyranosides as potential molecular probes for galactophilic proteins: assessment of monofluorogalactoside–LecA interactions S Fortin, D Lainé, C Bouzriba, D Giguère, E Shanina, V Denavit, É Gillon, ... VCH, 2019 | | 2019 |