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Andras Kotschy
Andras Kotschy
Servier Research Institute of Medicinal Chemistry
Verified email at servier.com
Title
Cited by
Cited by
Year
The MCL1 inhibitor S63845 is tolerable and effective in diverse cancer models
A Kotschy, Z Szlavik, J Murray, J Davidson, AL Maragno, ...
Nature 538 (7626), 477-482, 2016
9952016
Sonogashira coupling of aryl halides catalyzed by palladium on charcoal
Z Novák, A Szabó, J Répási, A Kotschy
The Journal of Organic Chemistry 68 (8), 3327-3329, 2003
2182003
Tandem Sonogashira coupling: An efficient tool for the synthesis of diarylalkynes
Z Novák, P Nemes, A Kotschy
Organic letters 6 (26), 4917-4920, 2004
1502004
Aromatic character of the benzene ring present in various topological environments in benzenoid hydrocarbons. Nonequivalence of indices of aromaticity
TM Krygowski, A Ciesielski, CW Bird, A Kotschy
Journal of chemical information and computer sciences 35 (2), 203-210, 1995
1481995
Modular synthesis of heterocyclic carbene precursors
A Paczal, AC Bényei, A Kotschy
The Journal of Organic Chemistry 71 (16), 5969-5979, 2006
1272006
Selective nucleophilic substitutions on tetrazines
Z Novak, B Bostai, M Csekei, KA Lorincz, A Kotschy
Heterocycles 60 (12), 2653-+, 2003
882003
First cross-coupling reactions on tetrazines
Z Novák, A Kotschy
Organic letters 5 (19), 3495-3497, 2003
872003
The chemistry behind ADCs
V Kostova, P Désos, JB Starck, A Kotschy
Pharmaceuticals 14 (5), 442, 2021
852021
Development of a one-pot sequential Sonogashira coupling for the synthesis of benzofurans
M Csékei, Z Novák, A Kotschy
Tetrahedron 64 (37), 8992-8996, 2008
722008
Small molecule glucokinase activators disturb lipid homeostasis and induce fatty liver in rodents: a warning for therapeutic applications in humans
F De Ceuninck, C Kargar, C Ilic, A Caliez, JO Rolin, T Umbdenstock, ...
British journal of pharmacology 168 (2), 339-353, 2013
712013
Efficient copper-catalyzed trifluoromethylation of aromatic and heteroaromatic iodides: The beneficial anchoring effect of borates
Z Gonda, S Kovacs, C Wéber, T Gáti, A Mészáros, A Kotschy, Z Novák
Organic letters 16 (16), 4268-4271, 2014
702014
The first total synthesis of Cicerfuran utilizing a one-pot synthesis of hydroxylated benzofurans
Z Novák, G Timári, A Kotschy
Tetrahedron 59 (38), 7509-7513, 2003
662003
Discovery of S64315, a potent and selective Mcl-1 inhibitor
Z Szlavik, M Csekei, A Paczal, ZB Szabo, S Sipos, G Radics, ...
Journal of Medicinal Chemistry 63 (22), 13762-13795, 2020
602020
Asymmetric synthesis in ionic liquids
A Paczal, A Kotschy
Monatshefte für Chemie-Chemical Monthly 138, 1115-1123, 2007
572007
Structure-guided discovery of a selective Mcl-1 inhibitor with cellular activity
Z Szlávik, L Ondi, M Csékei, A Paczal, ZB Szabó, G Radics, J Murray, ...
Journal of Medicinal Chemistry 62 (15), 6913-6924, 2019
562019
Sequential and domino Sonogashira coupling: Efficient tools for the synthesis of diarylalkynes
A Nagy, Z Novák, A Kotschy
Journal of organometallic chemistry 690 (20), 4453-4461, 2005
552005
Establishing drug discovery and identification of hit series for the anti-apoptotic proteins, Bcl-2 and Mcl-1
JB Murray, J Davidson, I Chen, B Davis, P Dokurno, CJ Graham, R Harris, ...
ACS omega 4 (5), 8892-8906, 2019
472019
Heterocycles from transition metal catalysis: formation and functionalization
A Kotschy, G Timári
Springer Science & Business Media, 2005
472005
The azaphilic addition of organometallic reagents on tetrazines: scope and limitations
J Faragó, Z Novák, G Schlosser, A Csámpai, A Kotschy
Tetrahedron 60 (9), 1991-1996, 2004
472004
Ethynyl-cyclohexanol: an efficient acetylene surrogate in Sonogashira coupling
M Csékei, Z Novák, A Kotschy
Tetrahedron 64 (6), 975-982, 2008
462008
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