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Eric Marsault
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Macrocycles are great cycles: applications, opportunities, and challenges of synthetic macrocycles in drug discovery
E Marsault, ML Peterson
Journal of medicinal chemistry 54 (7), 1961-2004, 2011
7372011
The transannular Diels-Alder strategy: applications to total synthesis
E Marsault, A Toró, P Nowak, P Deslongchamps
Tetrahedron 20 (57), 4243-4260, 2001
1592001
Tomatidine acts in synergy with aminoglycoside antibiotics against multiresistant Staphylococcus aureus and prevents virulence gene expression
G Mitchell, M Lafrance, S Boulanger, DL Séguin, I Guay, M Gattuso, ...
Journal of antimicrobial chemotherapy 67 (3), 559-568, 2012
1032012
Discovery and structure–activity relationship of a bioactive fragment of ELABELA that modulates vascular and cardiac functions
A Murza, X Sainsily, D Coquerel, J Côté, P Marx, É Besserer-Offroy, ...
Journal of medicinal chemistry 59 (7), 2962-2972, 2016
972016
Conjugation of a brain-penetrant peptide with neurotensin provides antinociceptive properties
M Demeule, N Beaudet, A Régina, É Besserer-Offroy, A Murza, ...
The Journal of clinical investigation 124 (3), 1199-1213, 2014
972014
Elucidation of the structure–activity relationships of apelin: influence of unnatural amino acids on binding, signaling, and plasma stability
A Murza, A Parent, E Besserer‐Offroy, H Tremblay, F Karadereye, ...
ChemMedChem 7 (2), 318-325, 2012
972012
Matriptase proteolytically activates influenza virus and promotes multicycle replication in the human airway epithelium
A Beaulieu, É Gravel, A Cloutier, I Marois, É Colombo, A Désilets, ...
Journal of virology 87 (8), 4237-4251, 2013
862013
Diversity-oriented synthesis: basics and applications in organic synthesis, drug discovery, and chemical biology
A Trabocchi
John Wiley & Sons, 2013
85*2013
Optimization of the potency and pharmacokinetic properties of a macrocyclic ghrelin receptor agonist (Part I): development of ulimorelin (TZP-101) from hit to clinic
HR Hoveyda, E Marsault, R Gagnon, AP Mathieu, M Vézina, A Landry, ...
Journal of medicinal chemistry 54 (24), 8305-8320, 2011
732011
Tomatidine inhibits replication of Staphylococcus aureus small-colony variants in cystic fibrosis airway epithelial cells
G Mitchell, M Gattuso, G Grondin, É Marsault, K Bouarab, F Malouin
Antimicrobial agents and chemotherapy 55 (5), 1937-1945, 2011
712011
Discovery of a new class of macrocyclic antagonists to the human motilin receptor
E Marsault, HR Hoveyda, ML Peterson, C Saint-Louis, A Landry, ...
Journal of medicinal chemistry 49 (24), 7190-7197, 2006
692006
Macrocyclic cell penetrating peptides: a study of structure-penetration properties
H Traboulsi, H Larkin, MA Bonin, L Volkov, CL Lavoie, E Marsault
Bioconjugate chemistry 26 (3), 405-411, 2015
682015
Design and synthesis of potent, selective inhibitors of matriptase
É Colombo, A Désilets, D Duchêne, F Chagnon, R Najmanovich, R Leduc, ...
ACS medicinal chemistry letters 3 (7), 530-534, 2012
672012
Stability and degradation patterns of chemically modified analogs of apelin‐13 in plasma and cerebrospinal fluid
A Murza, K Belleville, JM Longpré, P Sarret, É Marsault
Peptide Science 102 (4), 297-303, 2014
662014
Preparation of chiral phosphorothioate oligomers
G Just, Z Xin, E Marsault, Y Jin
US Patent 5,734,041, 1998
611998
Targeting matriptase in breast cancer abrogates tumour progression via impairment of stromal-epithelial growth factor signalling
GL Zoratti, LM Tanabe, FA Varela, AS Murray, C Bergum, É Colombo, ...
Nature communications 6 (1), 1-13, 2015
582015
Preparation of phosphorothioate and boranophosphate oligomers
G Just, Z Xin, E Marsault, Y Jin, J Wang, M Manoharan
US Patent 6,160,109, 2000
532000
Experimental treatment of Staphylococcus aureus bovine intramammary infection using a guanine riboswitch ligand analog
C Ster, M Allard, S Boulanger, ML Boulet, J Mulhbacher, DA Lafontaine, ...
Journal of dairy science 96 (2), 1000-1008, 2013
492013
Tomatidine is a lead antibiotic molecule that targets Staphylococcus aureus ATP synthase subunit C
M Lamontagne Boulet, C Isabelle, I Guay, E Brouillette, JP Langlois, ...
Antimicrobial agents and chemotherapy 62 (6), e02197-17, 2018
482018
C-Terminal modifications of apelin-13 significantly change ligand binding, receptor signaling, and hypotensive action
A Murza, E Besserer-Offroy, J Cote, P Berube, JM Longpre, R Dumaine, ...
Journal of medicinal chemistry 58 (5), 2431-2440, 2015
462015
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