A highly efficient in situ N-acetylation approach for solid phase synthesis K Chandra, TK Roy, JN Naoum, C Gilon, RB Gerber, A Friedler Organic & Biomolecular Chemistry 12 (12), 1879-1884, 2014 | 16 | 2014 |
DMAP-assisted sulfonylation as an efficient step for the methylation of primary amine motifs on solid support JN Naoum, K Chandra, D Shemesh, RB Gerber, C Gilon, M Hurevich Beilstein journal of organic chemistry 13 (1), 806-816, 2017 | 12 | 2017 |
Stirring peptide synthesis to a new level of efficiency JN Naoum, I Alshanski, G Mayer, P Strauss, M Hurevich Organic Process Research & Development 26 (1), 129-136, 2022 | 10 | 2022 |
Diffusion-enhanced amide bond formation on a solid support JN Naoum, I Alshanski, A Gitlin-Domagalska, M Bentolila, C Gilon, ... Organic Process Research & Development 23 (12), 2733-2739, 2019 | 9 | 2019 |
Mechanistic studies of malonic acid‐mediated in situ acylation K Chandra, JN Naoum, TK Roy, C Gilon, RB Gerber, A Friedler Peptide Science 104 (5), 495-505, 2015 | 4 | 2015 |
Synthesis and pharmacological characterization of Visabron, a backbone cyclic peptide dual antagonist of α4β1 (VLA-4)/α9β1 integrin for therapy of multiple sclerosis C Gilon, M Klazas, A Lahiani, A Schumacher-Klinger, S Merzbach, ... JACS Au 1 (12), 2361-2376, 2021 | 3 | 2021 |
Somatostatin prodrugs A Hoffman, C Gilon, A Klinger, J Naoum US Patent 11,261,215, 2022 | | 2022 |