| Prospective Evaluation of Free Energy Calculations for the Prioritization of Cathepsin L Inhibitors B Kuhn, M Tichý, L Wang, S Robinson, RE Martin, A Kuglstatter, J Benz, ... Journal of Medicinal Chemistry 60 (6), 2485-2497, 2017 | 130 | 2017 |
| Structural characterization of the highly cyclized lantibiotic paenicidin A via a partial desulfurization/reduction strategy CT Lohans, Z Huang, MJ van Belkum, M Giroud, CS Sit, EM Steels, ... Journal of the American Chemical Society 134 (48), 19540-19543, 2012 | 64 | 2012 |
| Inhibition of the Cysteine Protease Human Cathepsin L by Triazine Nitriles: Amide⋅⋅⋅ Heteroarene π‐Stacking Interactions and Chalcogen Bonding in the S3 Pocket M Giroud, J Ivkovic, M Martignoni, M Fleuti, N Trapp, W Haap, ... ChemMedChem 12 (3), 257-270, 2017 | 56 | 2017 |
| Arynes and Cyclic Alkynes as Synthetic Building Blocks for Stereodefined Quaternary Centers NKG E. N. Picazo, S. M. Anthony, M. Giroud, A. Simon, M. A. Miller, K. N. Houk J. Am. Chem. Soc. 140 (24), 7605-7610, 2018 | 48 | 2018 |
| 2H-1,2,3-Triazole-Based Dipeptidyl Nitriles: Potent, Selective, and Trypanocidal Rhodesain Inhibitors by Structure-Based Design M Giroud, B Kuhn, S Saint-Auret, C Kuratli, RE Martin, F Schuler, ... Journal of medicinal chemistry 61 (8), 3370-3388, 2018 | 48 | 2018 |
| Chemoenzymatic conversion of amides to enantioenriched alcohols in aqueous medium JE Dander, M Giroud, S Racine, ER Darzi, O Alvizo, D Entwistle, NK Garg Communications Chemistry 2 (1), 82, 2019 | 45 | 2019 |
| Fluorine Scan of Inhibitors of the Cysteine Protease Human Cathepsin L: Dipolar and Quadrupolar Effects in the π‐Stacking of Fluorinated Phenyl Rings on Peptide Amide Bonds M Giroud, M Harder, B Kuhn, W Haap, N Trapp, WB Schweizer, ... ChemMedChem 11 (10), 1042-1047, 2016 | 39 | 2016 |
| Repurposing a Library of Human Cathepsin L Ligands: Identification of Macrocyclic Lactams as Potent Rhodesain and Trypanosoma brucei Inhibitors M Giroud, U Dietzel, L Anselm, D Banner, A Kuglstatter, J Benz, JB Blanc, ... Journal of medicinal chemistry 61 (8), 3350-3369, 2018 | 36 | 2018 |
| Replacement of Water Molecules in a Phosphate Binding Site by Furanoside‐Appended lin‐Benzoguanine Ligands of tRNA‐Guanine Transglycosylase (TGT) LJ Barandun, FR Ehrmann, D Zimmerli, F Immekus, M Giroud, ... Chemistry-A European Journal 21 (1), 126-135, 2015 | 16 | 2015 |
| Trypanosomes inhibitors M Giroud, W Haap, B Kuhn, RE Martin US Patent 10,377,719, 2019 | 1 | 2019 |
| Arynes as synthetic building blocks for stereodefined quaternary centers M Giroud, N Garg ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 256, 2018 | | 2018 |
| N-Cyanocyclopropyl 2-Aminoalkanamides as Trypanosome Inhibitors and Their Preparation M Giroud, W Haap, B Kuhn, R Martin | | 2017 |
| The cysteine proteases human cathepsin L and rhodesain: investigation of the stacking of fluorinated arenes and heteroarenes on peptide amide bonds and the development of … M Giroud ETH Zurich, 2016 | | 2016 |
| Fluorine scan at the active sites of rhodesain and human cathepsin L: Enhanced binding affinity by stacking of fluorinated phenyl rings on flat dipeptide fragments M Giroud, M Harder, B Kuhn, W Haap, T Schirmeister, F Diederich ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 250, 2015 | | 2015 |
| Frontispiece: Replacement of Water Molecules in a Phosphate Binding Site by Furanoside‐Appended lin‐Benzoguanine Ligands of tRNA‐Guanine Transglycosylase (TGT) LJ Barandun, FR Ehrmann, D Zimmerli, F Immekus, M Giroud, ... Chemistry-A European Journal 21 (1), 2015 | | 2015 |
| Structural Characterization of Lantibiotic Paenicidin A via a Partial Desulfurization Approach CT Lohans, Z Huang, MJ van Belkum, M Giroud, CS Sit, JC Vederas BIOPOLYMERS 100 (3), 282-282, 2013 | | 2013 |
