Follow
Ewelina Węglarz-Tomczak
Ewelina Węglarz-Tomczak
CSO & Founder at NatInLab, Senior Research Scientist at HIMS University
Verified email at natinlab.com - Homepage
Title
Cited by
Cited by
Year
Azo dyes–biological activity and synthetic strategy
E Weglarz-Tomczak, L Gorecki
Chemik 66 (12), 1298-1307, 2012
792012
Identification of ebselen and its analogues as potent covalent inhibitors of papain-like protease from SARS-CoV-2
E Weglarz-Tomczak, JM Tomczak, M Talma, M Burda-Grabowska, ...
Scientific reports 11 (1), 3640, 2021
662021
Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases
S Vassiliou, E Weglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, ...
Journal of medicinal chemistry 57 (19), 8140-8151, 2014
512014
Ebselen as a highly active inhibitor of PLProCoV2
E Węglarz-Tomczak, JM Tomczak, M Talma, S Brul
BioRxiv, 2020.05. 17.100768, 2020
312020
Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and …
E Węglarz-Tomczak, M Burda-Grabowska, M Giurg, A Mucha
Bioorganic & Medicinal Chemistry Letters 26 (21), 5254-5259, 2016
312016
Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues
E Węglarz-Tomczak, S Vassiliou, A Mucha
Bioorganic & Medicinal Chemistry Letters 26 (16), 4122-4126, 2016
262016
A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases
E Węglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, A Joachimiak, ...
European journal of medicinal chemistry 117, 187-196, 2016
252016
Estimating kinetic constants in the Michaelis–Menten model from one enzymatic assay using Approximate Bayesian Computation
JM Tomczak, E Węglarz‐Tomczak
FEBS letters 593 (19), 2742-2750, 2019
232019
An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and …
E Węglarz-Tomczak, M Poręba, A Byzia, Ł Berlicki, B Nocek, R Mulligan, ...
Biochimie 95 (2), 419-428, 2013
232013
An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and …
E Węglarz-Tomczak, M Poręba, ...
Biochimie 95 (2), 419-428, 2013
232013
Controlling the Helix Handedness of ααβ‐Peptide Foldamers through Sequence Shifting
M Szefczyk, E Węglarz‐Tomczak, P Fortuna, A Krzysztoń, ...
Angewandte Chemie International Edition 56 (8), 2087-2091, 2017
162017
Discovery of potent inhibitors of PLproCoV2 by screening a library of selenium-containing compounds
E Węglarz-Tomczak, JM Tomczak, M Giurg, M Burda-Grabowska, S Brul
bioRxiv, 2020.05. 20.107052, 2020
122020
Differential evolution with reversible linear transformations
JM Tomczak, E Węglarz-Tomczak, AE Eiben
Proceedings of the 2020 Genetic and Evolutionary Computation Conference …, 2020
112020
Deep learning and transfer learning for automatic cell counting in microscope images of human cancer cell lines
F Lavitt, DJ Rijlaarsdam, D van der Linden, E Weglarz-Tomczak, ...
Applied Sciences 11 (11), 4912, 2021
92021
Neutral metalloaminopeptidases APN and MetAP2 as newly discovered anticancer molecular targets of actinomycin D and its simple analogs
E Węglarz-Tomczak, M Talma, M Giurg, HV Westerhoff, R Janowsk, ...
Oncotarget 9 (50), 29365-29378, 2018
92018
Helix-loop-helix peptide foldamers and their use in the construction of hydrolase mimetics
M Drewniak, E Węglarz-Tomczak, K Ożga, E Rudzińska-Szostak, ...
Bioorganic Chemistry 81, 356-361, 2018
82018
Simultaneous integration of gene expression and nutrient availability for studying the metabolism of hepatocellular carcinoma cell lines
E Weglarz-Tomczak, TDGA Mondeel, DGE Piebes, HV Westerhoff
Biomolecules 11 (4), 490, 2021
52021
Enantiomeric α, β-diaminoethylphosphonic acids as potent inhibitors of aminopeptidases—stereoselective synthesis and biological activity
E Węglarz-Tomczak, K Staszewska, M Talma, A Mucha
Tetrahedron Letters 57 (43), 4812-4814, 2016
52016
GEM-based metabolic profiling for human bone osteosarcoma under different glucose and glutamine availability
E Weglarz-Tomczak, DJ Rijlaarsdam, JM Tomczak, S Brul
International Journal of Molecular Sciences 22 (3), 1470, 2021
32021
Barwniki azowe–aktywność biologiczna i strategie syntezy
E Węglarz-Tomczak, Ł Górecki
Chemik 66 (12), 1298-1302, 2012
32012
The system can't perform the operation now. Try again later.
Articles 1–20