| Azo dyes–biological activity and synthetic strategy E Weglarz-Tomczak, L Gorecki Chemik 66 (12), 1298-1307, 2012 | 79 | 2012 |
| Identification of ebselen and its analogues as potent covalent inhibitors of papain-like protease from SARS-CoV-2 E Weglarz-Tomczak, JM Tomczak, M Talma, M Burda-Grabowska, ... Scientific reports 11 (1), 3640, 2021 | 66 | 2021 |
| Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases S Vassiliou, E Weglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, ... Journal of medicinal chemistry 57 (19), 8140-8151, 2014 | 51 | 2014 |
| Ebselen as a highly active inhibitor of PLProCoV2 E Węglarz-Tomczak, JM Tomczak, M Talma, S Brul BioRxiv, 2020.05. 17.100768, 2020 | 31 | 2020 |
| Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and … E Węglarz-Tomczak, M Burda-Grabowska, M Giurg, A Mucha Bioorganic & Medicinal Chemistry Letters 26 (21), 5254-5259, 2016 | 31 | 2016 |
| Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues E Węglarz-Tomczak, S Vassiliou, A Mucha Bioorganic & Medicinal Chemistry Letters 26 (16), 4122-4126, 2016 | 26 | 2016 |
| A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases E Węglarz-Tomczak, Ł Berlicki, M Pawełczak, B Nocek, A Joachimiak, ... European journal of medicinal chemistry 117, 187-196, 2016 | 25 | 2016 |
| Estimating kinetic constants in the Michaelis–Menten model from one enzymatic assay using Approximate Bayesian Computation JM Tomczak, E Węglarz‐Tomczak FEBS letters 593 (19), 2742-2750, 2019 | 23 | 2019 |
| An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and … E Węglarz-Tomczak, M Poręba, A Byzia, Ł Berlicki, B Nocek, R Mulligan, ... Biochimie 95 (2), 419-428, 2013 | 23 | 2013 |
| An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and … E Węglarz-Tomczak, M Poręba, ... Biochimie 95 (2), 419-428, 2013 | 23 | 2013 |
| Controlling the Helix Handedness of ααβ‐Peptide Foldamers through Sequence Shifting M Szefczyk, E Węglarz‐Tomczak, P Fortuna, A Krzysztoń, ... Angewandte Chemie International Edition 56 (8), 2087-2091, 2017 | 16 | 2017 |
| Discovery of potent inhibitors of PLproCoV2 by screening a library of selenium-containing compounds E Węglarz-Tomczak, JM Tomczak, M Giurg, M Burda-Grabowska, S Brul bioRxiv, 2020.05. 20.107052, 2020 | 12 | 2020 |
| Differential evolution with reversible linear transformations JM Tomczak, E Węglarz-Tomczak, AE Eiben Proceedings of the 2020 Genetic and Evolutionary Computation Conference …, 2020 | 11 | 2020 |
| Deep learning and transfer learning for automatic cell counting in microscope images of human cancer cell lines F Lavitt, DJ Rijlaarsdam, D van der Linden, E Weglarz-Tomczak, ... Applied Sciences 11 (11), 4912, 2021 | 9 | 2021 |
| Neutral metalloaminopeptidases APN and MetAP2 as newly discovered anticancer molecular targets of actinomycin D and its simple analogs E Węglarz-Tomczak, M Talma, M Giurg, HV Westerhoff, R Janowsk, ... Oncotarget 9 (50), 29365-29378, 2018 | 9 | 2018 |
| Helix-loop-helix peptide foldamers and their use in the construction of hydrolase mimetics M Drewniak, E Węglarz-Tomczak, K Ożga, E Rudzińska-Szostak, ... Bioorganic Chemistry 81, 356-361, 2018 | 8 | 2018 |
| Simultaneous integration of gene expression and nutrient availability for studying the metabolism of hepatocellular carcinoma cell lines E Weglarz-Tomczak, TDGA Mondeel, DGE Piebes, HV Westerhoff Biomolecules 11 (4), 490, 2021 | 5 | 2021 |
| Enantiomeric α, β-diaminoethylphosphonic acids as potent inhibitors of aminopeptidases—stereoselective synthesis and biological activity E Węglarz-Tomczak, K Staszewska, M Talma, A Mucha Tetrahedron Letters 57 (43), 4812-4814, 2016 | 5 | 2016 |
| GEM-based metabolic profiling for human bone osteosarcoma under different glucose and glutamine availability E Weglarz-Tomczak, DJ Rijlaarsdam, JM Tomczak, S Brul International Journal of Molecular Sciences 22 (3), 1470, 2021 | 3 | 2021 |
| Barwniki azowe–aktywność biologiczna i strategie syntezy E Węglarz-Tomczak, Ł Górecki Chemik 66 (12), 1298-1302, 2012 | 3 | 2012 |
Jakub M. TomczakAssistant Professor at Vrije Universiteit AmsterdamVerified email at vu.nl
